1. Vías de señalización
  2. GPCR/G Protein
  3. P2Y Receptor
  4. P2Y12 Receptor Isoform
  5. P2Y12 Receptor Activator

P2Y12 Receptor Activator

P2Y12 Receptor Activators (2):

Cat. No. Nombre del producto Efecto Pureza
  • HY-107752A
    2-(Phenylethynyl)-ATP ammonium
    Activator
    2-(Phenylethynyl)-ATP (ammonium) is a selective and potent GPR17 agonist with an EC50 of 35 pM. 2-(Phenylethynyl)-ATP (ammonium) also shows weak activation of P2Y Receptor. 2-(Phenylethynyl)-ATP (ammonium) can be used for the research of neurological disease.
  • HY-134353B
    ADP-β-S trilithium
    Activator
    ADP-β-S (Adenosine 5'-(β-thiodiphosphate)) trilithium is a non-hydrolyzable ADP analog and a P2Y12 receptor agonist. ADP-β-S trilithium activates the P2Y12 receptor in microglia, thereby triggering downstream inflammatory signaling pathways. ADP-β-S trilithium activates P2Y purinergic receptors in rat pancreatic β cells and enhances glucose-induced insulin secretion. ADP-β-S trilithium can be used in the research of diseases such as inflammation and diabetes.