ARTD10/PARP10-IN-1
ARTD10/PARP10-IN-1 (compound 23) is a potent and non-selective PARP inhibitor, targeting to mono-ADP-ribosyltransferases ARTD7/PARP15, ARTD8/PARP14, ARTD10/PARP10 and poly(ADP-ribose) polymerase-1 (ARTD1/PARP1) with IC50s of 1.7 μM, 1.6 μM, 0.8 μM, and 4.4 μM, respectively.
For research use only. We do not sell to patients.
- CAS No.: 1708103-76-7
- Formula: C12H12N2O4
- Molecular Weight:248.23
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
ARTD1/PARP1 4.4 μM (IC50) |
ARTD10/PARP10 0.8 μM (IC50) |
ARTD8/PARP14 1.6 μM (IC50) |
ARTD7/PARP15 1.7 μM (IC50) |
Chemical Information
-
CAS No. 1708103-76-7
-
Molecular Weight 248.23
-
Formula C12H12N2O4
-
SMILES
COC(/C=C\C(NC1=CC(C(N)=O)=CC=C1)=O)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)