BCFTP
BCFTP is a potent, orally active and selective human Mas-related G protein-coupled receptor X1 (MrgprX1)-positive allosteric modulator. BCFTP selectively potentiates MrgprX1 signaling in HEK293 cells. BCFTP alleviates specific neuropathic pain-related behaviors in a humanized MrgprX1 mouse model of chronic constrictive injury (CCI) in a MrgprX1-dependent manner. BCFTP synergistically enhances psychoactive substances analgesia in CCI MrgprX1 mice. BCFTP can be used for neuropathic pain research.
For research use only. We do not sell to patients.
- CAS No.: 2781215-95-8
- Formula: C23H17ClF4N2O2S
- Molecular Weight:496.90
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 2781215-95-8
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Molecular Weight 496.90
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Formula C23H17ClF4N2O2S
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SMILES
CC(C)(C)C1=C(C2=CC=C(Cl)C=C2)C3=C(S1)N=CN=C3OC4=C(F)C=CC=C4OC(F)(F)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)