130736-25-3
130736-25-3
Chemical Structure
U 84569
- CAS No.: 130736-25-3
- Formula:C25H23NO4
- Molecular Weight:401.45
InChIKey: GZIQMRPAMVVPAK-UHFFFAOYSA-N
SMILES: O=C1C=C(N2CCOCC2)OC3=C(C)C(OCC4=CC=CC5=C4C=CC=C5)=CC=C31
Biological Activity: U 84569 is a potent low-Km cAMP-dependent Phosphodiesterase inhibitor, with an IC50 value of 300 nM in platelet cytosol. By inhibiting phosphodiesterase and elevating cAMP levels, U 84569 indirectly blocks receptor-mediated Phospholipase C activation, thereby inhibiting platelet aggregation[1].
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U 84569 | U 84569 is a potent low-Km cAMP-dependent Phosphodiesterase inhibitor, with an IC50 value of 300 nM in platelet cytosol. By inhibiting phosphodiesterase and elevating cAMP levels, U 84569 indirectly blocks receptor-mediated Phospholipase C activation, thereby inhibiting platelet aggregation. | |||||||||||||||||||||
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