1335138-89-0
Chemical Structure
DS-1040 Tosylate
- CAS No.: 1335138-89-0
- Formula:C23H35N3O5S
- Molecular Weight:465.61
IUPAC Name: (S)-5-amino-2-((1-((1r,4S)-4-methylcyclohexyl)-1H-imidazol-4-yl)methyl)pentanoic acid compound with 4-methylbenzenesulfonic acid (1:1)
InChIKey: BEUWOXSXOMMLGF-HZPCBCDKSA-N
SMILES: O=C(O)[C@H](CC1=CN([C@H]2CC[C@H](C)CC2)C=N1)CCCN.CC3=CC=C(S(=O)(O)=O)C=C3
Biological Activity: DS-1040 Tosylate is an orally active, selective inhibitor of activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50s of 5.92 nM and 8.01 nM for human and rat TAFIa. DS-1040 Tosylate is a fibrinolysis enhancer for thromboembolic diseases[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DS-1040 Tosylate | 99.26% | DS-1040 Tosylate is an orally active, selective inhibitor of activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50s of 5.92 nM and 8.01 nM for human and rat TAFIa. DS-1040 Tosylate is a fibrinolysis enhancer for thromboembolic diseases. | ||||||||||||||||||||
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DS-1040 Tosylate (Standard) | ≥98% | DS-1040 Tosylate (Standard) is the analytical standard of DS-1040 Tosylate (HY-101918). This product is intended for research and analytical applications. DS-1040 Tosylate is an orally active, selective inhibitor of activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50s of 5.92 nM and 8.01 nM for human and rat TAFIa. DS-1040 Tosylate is a fibrinolysis enhancer for thromboembolic diseases. | ||||||||||||||||||||
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Similarity Score 0.74
HY-117745DS-1040 -
Similarity Score 0.62
HY-179636DS-1040 Tosylate prodrug-1 -
Similarity Score 0.52
HY-122052UK‑396082 -
Similarity Score 0.50
HY-168450trans-Cyclohexane-p-bis(C-OTs) -
Similarity Score 0.49
HY-1588054-Methoxy-α-pyrrolidinopropiophenone tosylate -
Similarity Score 0.48
HY-W002303L-Leucine benzyl ester p-toluenesulfonate -
Similarity Score 0.48
HY-W011200H-Gly-OBzl.TosOH -
Similarity Score 0.48
HY-W779904H-Gly-OBzl.TosOH-13C2,15N -
Similarity Score 0.48
HY-W765357Glycine-13C2,15N p-Toluenesulfonate -
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