1356497-92-1
1356497-92-1
Chemical Structure
PT-S58
- CAS No.: 1356497-92-1
- Formula:C17H22N2O5S2
- Molecular Weight:398.50
IUPAC Name: methyl 3-(N-(4-(tert-butylamino)-2-methoxyphenyl)sulfamoyl)thiophene-2-carboxylate
InChIKey: JSUWAIOZKBYWCJ-UHFFFAOYSA-N
SMILES: O=C(C1=C(S(=O)(NC2=CC=C(NC(C)(C)C)C=C2OC)=O)C=CS1)OC
Biological Activity: PT-S58, a GSK0660 derivative, is a PPARβ/δ full antagonist with an IC50 value of 98 nM. PT-S58 inhibits the agonist-induced transcriptional activity of PPARβ/δ in vitro[1].
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PT-S58 | PT-S58, a GSK0660 derivative, is a PPARβ/δ full antagonist with an IC50 value of 98 nM. PT-S58 inhibits the agonist-induced transcriptional activity of PPARβ/δ in vitro. | |||||||||||||||||||||
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