144231-85-6
Chemical Structure
Calpain-2-IN-1
- CAS No.: 144231-85-6
- Formula:C28H37N3O7
- Molecular Weight:527.61
IUPAC Name: benzyl ((S)-1-(((S)-1-((3,5-dimethoxybenzyl)amino)-1,2-dioxopentan-3-yl)amino)-4-methyl-1-oxopentan-2-yl)carbamate
InChIKey: ZPKXXXUPXHNDFV-ZEQRLZLVSA-N
SMILES: O=C(OCC1=CC=CC=C1)N[C@@H](CC(C)C)C(N[C@@H](CC)C(C(NCC2=CC(OC)=CC(OC)=C2)=O)=O)=O
Biological Activity: Calpain-2-IN-1 (Formula 1A) is a isoform-specific calpain-2 inhibitor with Kis of 181 nM and 7.8 nM for calpain-1, and calpain-2, respectively. Calpain-2-IN-1 can be used for the research of neurodegenerative diseases and other diseases of synaptic function[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Calpain-2-IN-1 | 98.05% | Calpain-2-IN-1 (Formula 1A) is a isoform-specific calpain-2 inhibitor with Kis of 181 nM and 7.8 nM for calpain-1, and calpain-2, respectively. Calpain-2-IN-1 can be used for the research of neurodegenerative diseases and other diseases of synaptic function. | ||||||||||||||||||||
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