1688684-07-2
Chemical Structure
MPX-004
- CAS No.: 1688684-07-2
- Formula:C17H15ClFN5O3S2
- Molecular Weight:455.91
IUPAC Name: 5-(((3-chloro-4-fluorophenyl)sulfonamido)methyl)-N-((2-methylthiazol-5-yl)methyl)pyrazine-2-carboxamide
InChIKey: BRNKHERDLJYUNK-UHFFFAOYSA-N
SMILES: O=C(C1=NC=C(CNS(=O)(C2=CC=C(C(Cl)=C2)F)=O)N=C1)NCC3=CN=C(C)S3
Biological Activity:
MPX-004 is a potent GluN2A antagonist. MPX-004 inhibits GluN2A-containing NMDA receptors expressed in HEK cells with an IC50 of 79 nM. MPX-004 has no inhibitory effect on GluN2B or GluN2D receptor-mediated responses. MPX-004 has the potential for neuropsychiatric and developmental disorders research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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MPX-004 | 99.58% | MPX-004 is a potent GluN2A antagonist. MPX-004 inhibits GluN2A-containing NMDA receptors expressed in HEK cells with an IC50 of 79 nM. MPX-004 has no inhibitory effect on GluN2B or GluN2D receptor-mediated responses. MPX-004 has the potential for neuropsychiatric and developmental disorders research. |
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Keywords
