186371-96-0
Chemical Structure
ZK168281
- CAS No.: 186371-96-0
- Formula:C32H46O5
- Molecular Weight:510.70
IUPAC Name: ethyl (E)-3-(1-((1R,4R,E)-4-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)-3,5-dihydroxy-2-methylenecyclohexylidene)ethylidene)-7a-methyloctahydro-1H-inden-1-yl)-1-hydroxypent-2-en-1-yl)cyclopropyl)acrylate
InChIKey: FUDAEUIGIJZUAY-UMIRZPQISA-N
SMILES: O=C(OCC)/C=C/C1([C@H](O)/C=C/[C@H]([C@H]2CC[C@@]3([H])/C(CCC[C@]23C)=C/C=C4C([C@@H](O)C[C@H](O)C\4)=C)C)CC1
Biological Activity: ZK168281 is a 25-carboxylic ester 1α,25(OH)2D3 analog and a pure VDR antagonist with a Kd value of 0.1 nM. ZK168281 is an effective inhibitor of the coactivator (CoA) interaction of its receptor[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ZK168281 | 98.0% | ZK168281 is a 25-carboxylic ester 1α,25(OH)2D3 analog and a pure VDR antagonist with a Kd value of 0.1 nM. ZK168281 is an effective inhibitor of the coactivator (CoA) interaction of its receptor. | ||||||||||||||||||||
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Keywords
