190328-44-0
190328-44-0
Chemical Structure
GR 128107
- CAS No.: 190328-44-0
- Formula:C16H20N2O2
- Molecular Weight:272.34
IUPAC Name: 1-(3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)ethan-1-one
InChIKey: RBINAFTXZHPTNU-UHFFFAOYSA-N
SMILES: CC(N1CC(CCC1)C2=CNC3=C2C=C(C=C3)OC)=O
Biological Activity: GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6)[1].
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GR 128107 | GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6). | |||||||||||||||||||||
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References
- [1]. Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75. [Content Brief]
Keywords
