GR 128107
GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6).
For research use only. We do not sell to patients.
- CAS No.: 190328-44-0
- Formula: C16H20N2O2
- Molecular Weight:272.34
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 190328-44-0
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Molecular Weight 272.34
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Formula C16H20N2O2
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SMILES
CC(N1CC(CCC1)C2=CNC3=C2C=C(C=C3)OC)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)