2259641-59-1
Chemical Structure
Ep300/CREBBP-IN-2
- CAS No.: 2259641-59-1
- Formula:C26H27F3N4O4
- Molecular Weight:516.51
IUPAC Name: (2R,4R)-1-(4,4-difluoro-1-(4-methoxyphenyl)cyclohexane-1-carbonyl)-4-fluoro-N-(2-oxo-2,3-dihydro-1H-pyrrolo[3,2-b]pyridin-5-yl)pyrrolidine-2-carboxamide
InChIKey: CVCCDDXWAXREGK-OXQOHEQNSA-N
SMILES: O=C([C@@H]1N(C(C2(C3=CC=C(OC)C=C3)CCC(F)(F)CC2)=O)C[C@H](F)C1)NC4=CC=C(NC(C5)=O)C5=N4
Biological Activity: Ep300/CREBBP-IN-2 (Example 73) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.052 and 0.148 μM, respectively. Ep300/CREBBP-IN-2 can be used for the research of cancer[1].
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Ep300/CREBBP-IN-2 | Ep300/CREBBP-IN-2 (Example 73) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.052 and 0.148 μM, respectively. Ep300/CREBBP-IN-2 can be used for the research of cancer. | |||||||||||||||||||||
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Keywords
