2322293-83-2
2322293-83-2
Chemical Structure
PI3Kα-IN-4
- CAS No.: 2322293-83-2
- Formula:C25H23ClFN5O5S
- Molecular Weight:560.00
IUPAC Name: (R)-3-(6-(5-((2-chloro-4-fluorophenyl)sulfonamido)-6-methoxypyridin-3-yl)-4-oxoquinazolin-3(4H)-yl)-N,2-dimethylpropanamide
InChIKey: LPATWVFSBNDSHR-CQSZACIVSA-N
SMILES: O=C(NC)[C@H](C)CN1C=NC2=C(C=C(C3=CC(NS(=O)(C4=CC=C(F)C=C4Cl)=O)=C(OC)N=C3)C=C2)C1=O
Biological Activity: PI3Kα-IN-4 is a potent, selective and orally active inhibitor of PI3Kα, with an IC50 of 1.8 nM. PI3Kα-IN-4 has antitumor activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PI3Kα-IN-4 | 99.76% | PI3Kα-IN-4 is a potent, selective and orally active inhibitor of PI3Kα, with an IC50 of 1.8 nM. PI3Kα-IN-4 has antitumor activity. | ||||||||||||||||||||
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References
Keywords
