2355304-05-9
2355304-05-9
Chemical Structure
RGH-122
- CAS No.: 2355304-05-9
- Formula:C24H25ClN4O3
- Molecular Weight:452.93
InChIKey: LFXCGLFTXRJJLT-RUCARUNLSA-N
SMILES: ClC1=CC=[C@]2[N@]3C([C@H](CC4)CC[C@@H]4OC5=NC=CC=C5)=NN=C3CC6(OCCO6)CC2=C1
Biological Activity: RGH-122 (compound 43) is an orally active, potent, selective, and hV1a receptor antagonist with Ki value of 0.3 nM and IC50 of 0.9 nM. RGH-122 showes microsomal stability with CLint value of 13/28/25 μL/min/mg[1].
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RGH-122 | RGH-122 (compound 43) is an orally active, potent, selective, and hV1a receptor antagonist with Ki value of 0.3 nM and IC50 of 0.9 nM. RGH-122 showes microsomal stability with CLint value of 13/28/25 μL/min/mg. | |||||||||||||||||||||
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References
Keywords
