2379279-96-4
Chemical Structure
HSD1590
- CAS No.: 2379279-96-4
- Formula:C20H18BN3O3
- Molecular Weight:359.19
IUPAC Name: (2-methoxy-3-(3,8,9,10-tetrahydrocyclopenta[c]pyrazolo[4,3-f]quinolin-7-yl)phenyl)boronic acid
InChIKey: WTZMCUOBQPTERK-UHFFFAOYSA-N
SMILES: COC(C(B(O)O)=CC=C1)=C1C(C2=C3CCC2)=NC4=C3C(C=NN5)=C5C=C4
Biological Activity: HSD1590 is potent ROCK inhibitor, with IC50s of 1.22 and 0.51 nM for ROCK1 and ROCK2, respectively. HSD1590 exhibits single digit nanomolar binding to ROCK (Kds<2 nM). HSD1590 displays low cytotoxicity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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HSD1590 | 99.00% | HSD1590 is potent ROCK inhibitor, with IC50s of 1.22 and 0.51 nM for ROCK1 and ROCK2, respectively. HSD1590 exhibits single digit nanomolar binding to ROCK (Kds<2 nM). HSD1590 displays low cytotoxicity. | ||||||||||||||||||||
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Keywords