2379409-91-1
Chemical Structure
CBP/p300-IN-15
- CAS No.: 2379409-91-1
- Formula:C26H28N4O5
- Molecular Weight:476.52
IUPAC Name: 1-methyl-3-((R)-3'-(2-((R)-3-methyl-1,3,4,5-tetrahydro-2H-benzo[c]azepin-2-yl)-2-oxoethyl)-2',4'-dioxo-2,3-dihydrospiro[indene-1,5'-oxazolidin]-5-yl)urea
InChIKey: VDINOEOOUILKFN-AKJBCIBTSA-N
SMILES: CNC(NC1=CC=C2C(CC[C@@]23OC(N(C3=O)CC(N4CC5=CC=CC=C5CC[C@H]4C)=O)=O)=C1)=O
Biological Activity: CBP/p300-IN-15 (compound 13a) is a potent p300/CBP inhibitor, with IC50 values of 2.50 and 28.0 nM, respectively. CBP/p300-IN-15 shows good activity against OVCAR-3 and A2780 cell line, with EC50 values of 0.865 and 2.71 μM, respectively. CBP/p300-IN-15 can be used for ovarian cancer research[1].
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CBP/p300-IN-15 | CBP/p300-IN-15 (compound 13a) is a potent p300/CBP inhibitor, with IC50 values of 2.50 and 28.0 nM, respectively. CBP/p300-IN-15 shows good activity against OVCAR-3 and A2780 cell line, with EC50 values of 0.865 and 2.71 μM, respectively. CBP/p300-IN-15 can be used for ovarian cancer research. | |||||||||||||||||||||
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Keywords
