245747-08-4
Chemical Structure
Pyr6
Synonym(s): N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide
- CAS No.: 245747-08-4
- Formula:C17H9F7N4O
- Molecular Weight:418.27
IUPAC Name: N-(4-(3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl)phenyl)-3-fluoroisonicotinamide
InChIKey: XZIQSOZOLJJMFN-UHFFFAOYSA-N
SMILES: O=C(C1=C(F)C=NC=C1)NC2=CC=C(N3N=C(C(F)(F)F)C=C3C(F)(F)F)C=C2
Biological Activity: Pyr6 is a selective store operated calcium entry (SOCE) inhibitor with an IC50 of 0.49 μM. Pyr6 displays 37-fold higher potency for RBL SOCE than for TRPC3 ROCE[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Pyr6 | 98.61% | Pyr6 is a selective store operated calcium entry (SOCE) inhibitor with an IC50 of 0.49 μM. Pyr6 displays 37-fold higher potency for RBL SOCE than for TRPC3 ROCE. | ||||||||||||||||||||
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Keywords