2654075-94-0
2654075-94-0
Chemical Structure
CDK7/12-IN-1
- CAS No.: 2654075-94-0
- Formula:C25H34N8O
- Molecular Weight:462.59
IUPAC Name: (3R,4R)-4-(((7-(((2,7-dimethylimidazo[1,2-a]pyridin-3-yl)methyl)amino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)methyl)piperidin-3-ol
InChIKey: IHXKZRXUGKSPTO-NQIIRXRSSA-N
SMILES: O[C@H]1CNCC[C@@H]1CNC2=NC3=C(C(C)C)C=NN3C(NCC4=C(C)N=C5C=C(C)C=CN54)=C2
Biological Activity: CDK7/12-IN-1 is a selective CDK7/12 inhibitor with IC50s of 3 and 277 nM for CDK7 and CDK 12, respectively. CDK7 and CDK12 inhibition is an effective strategy to inhibit tumour growth[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CDK7/12-IN-1 | 99.66% | CDK7/12-IN-1 is a selective CDK7/12 inhibitor with IC50s of 3 and 277 nM for CDK7 and CDK 12, respectively. CDK7 and CDK12 inhibition is an effective strategy to inhibit tumour growth. | ||||||||||||||||||||
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References
Keywords
