2819989-68-7
2819989-68-7
Chemical Structure
PBRM1-BD2-IN-7
- CAS No.: 2819989-68-7
- Formula:C16H15ClN2O
- Molecular Weight:286.76
IUPAC Name: N-((S)-1-(2-((R)-2-chloro-2-fluoroacetyl)-2-(((S)-2-oxopyrrolidin-3-yl)methyl)hydrazinyl)-4-methyl-1-oxopentan-2-yl)-4-fluoro-1H-indole-2-carboxamide
InChIKey: OKLYBCNMVQMCRF-UHFFFAOYSA-N
SMILES: O=C1NC(C2=C(C)C=CC=C2C)NC3=C1C(Cl)=CC=C3
Biological Activity: PBRM1-BD2-IN-7 is a selective and cell-active polybromo-1 (PBRM1) bromodomain inhibitor. PBRM1-BD2-IN-7 has inhibitory activity for PBRM1-BD2 with an IC50 value of 0.29 μM. PBRM1-BD2-IN-7 can be used for the research of cancer[1].
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PBRM1-BD2-IN-7 | PBRM1-BD2-IN-7 is a selective and cell-active polybromo-1 (PBRM1) bromodomain inhibitor. PBRM1-BD2-IN-7 has inhibitory activity for PBRM1-BD2 with an IC50 value of 0.29 μM. PBRM1-BD2-IN-7 can be used for the research of cancer. | |||||||||||||||||||||
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Keywords
