3031486-11-7
Chemical Structure
DNA Gyrase-IN-1
- CAS No.: 3031486-11-7
- Formula:C24H24FN7O6
- Molecular Weight:525.49
IUPAC Name: (2R,4S,4aS)-11-fluoro-2,4-dimethyl-2',4',6'-trioxo-8-(((S)-5-oxopyrrolidin-2-yl)methoxy)-1,1',2,3',4,4a,4',6'-octahydro-2'H,3H,6H-spiro[isoxazolo[4,5-g]pyrazino[1,2-a]quinoline-5,5'-pyrimidine]-3-carbonitrile
InChIKey: CEVFXBOLWXVYCW-FNPAYESESA-N
SMILES: C[C@@H]1N([C@@H](CN2C3=C(C4=C(C=C3CC5([C@]21[H])C(NC(NC5=O)=O)=O)C(OC[C@H]6NC(CC6)=O)=NO4)F)C)C#N
Biological Activity: DNA Gyrase-IN-1 (compound 42) is a potent and selective DNA gyrase inhibitor with an IC50 value of 2.6 µM. DNA Gyrase-IN-1 has high inhibitory activity against Mycobacterium tuberculosis (Mtb) with MIC of 0.49 µM. DNA Gyrase-IN-1 can be used for researching tuberculosis[1].
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DNA Gyrase-IN-1 | DNA Gyrase-IN-1 (compound 42) is a potent and selective DNA gyrase inhibitor with an IC50 value of 2.6 µM. DNA Gyrase-IN-1 has high inhibitory activity against Mycobacterium tuberculosis (Mtb) with MIC of 0.49 µM. DNA Gyrase-IN-1 can be used for researching tuberculosis. | |||||||||||||||||||||
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Keywords
