3139993-34-0
3139993-34-0
Chemical Structure
Sigma ligand-2
- CAS No.: 3139993-34-0
- Formula:C20H24N2O
- Molecular Weight:308.42
InChIKey: OFQPZGYARCLOLC-OYKVQYDMSA-N
SMILES: CC(C)C(C1=CC=CC=C1)NC([C@@H]2CC3=CC=CC=C3CN2)=O
Biological Activity: Sigma ligand-2 is a sigma-1 receptor (σ1R) ligand with high-affinity binding and selectivity over the sigma-2 receptor (σ2R). Sigma ligand-2 binds σ1R with a Ki of 7.01 nM. Sigma ligand-2 shows negligible σ2R binding and a σ2R Ki of >10,000 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Sigma ligand-2 | Sigma ligand-2 is a sigma-1 receptor (σ1R) ligand with high-affinity binding and selectivity over the sigma-2 receptor (σ2R). Sigma ligand-2 binds σ1R with a Ki of 7.01 nM. Sigma ligand-2 shows negligible σ2R binding and a σ2R Ki of >10,000 nM. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
