Sigma ligand-2
Sigma ligand-2 is a sigma-1 receptor (σ1R) ligand with high-affinity binding and selectivity over the sigma-2 receptor (σ2R). Sigma ligand-2 binds σ1R with a Ki of 7.01 nM. Sigma ligand-2 shows negligible σ2R binding and a σ2R Ki of >10,000 nM.
For research use only. We do not sell to patients.
- CAS No.: 3139993-34-0
- Formula: C20H24N2O
- Molecular Weight:308.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
Description
IC50 & Target
[1]|
σ1R 7.01 nM (Ki) |
Sigma 2 Receptor > 10,000 nM (Ki) |
In Vitro
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3139993-34-0
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Molecular Weight 308.42
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Formula C20H24N2O
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SMILES
CC(C)C(C1=CC=CC=C1)NC([C@@H]2CC3=CC=CC=C3CN2)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Sigma ligand-2 Related Classifications
HY-190678 Related Classifications
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