36840-10-5
36840-10-5
Chemical Structure
LPA2 antagonist 2
- CAS No.: 36840-10-5
- Formula:C20H16N2O6
- Molecular Weight:380.35
IUPAC Name: (2E,2'E)-4,4'-([1,1'-biphenyl]-4,4'-diylbis(azanediyl))bis(4-oxobut-2-enoic acid)
InChIKey: FTLRWRKPUWMOMS-WGDLNXRISA-N
SMILES: O=C(O)/C=C/C(NC1=CC=C(C2=CC=C(NC(/C=C/C(O)=O)=O)C=C2)C=C1)=O
Biological Activity: LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM. LPA2 antagonist 2 is >480-fold more selective than LPA3 (IC50 of 13.85 μM)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
LPA2 antagonist 2 | 95.0% | LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM. LPA2 antagonist 2 is >480-fold more selective than LPA3 (IC50 of 13.85 μM). | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
