396129-53-6
396129-53-6
Chemical Structure
LY-364947
Synonym(s): HTS466284
- CAS No.: 396129-53-6
- Formula:C17H12N4
- Molecular Weight:272.30
IUPAC Name: 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)quinoline
InChIKey: IBCXZJCWDGCXQT-UHFFFAOYSA-N
SMILES: C1(C2=CNN=C2C3=NC=CC=C3)=CC=NC4=CC=CC=C14
Biological Activity: LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM, and exhibits 7-fold selectivity over TGFβR-II[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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LY-364947 | 99.23% | LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM, and exhibits 7-fold selectivity over TGFβR-II. | ||||||||||||||||||||
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References
Keywords
