879368-27-1
879368-27-1
Chemical Structure
H3R antagonist 5
- CAS No.: 879368-27-1
- Formula:C23H32N2O4
- Molecular Weight:400.51
IUPAC Name: (1r,4r)-5'-methoxy-N-methyl-3'-oxo-N-(2-(piperidin-1-yl)ethyl)-3'H-spiro[cyclohexane-1,1'-isobenzofuran]-4-carboxamide
InChIKey: AEWLECDUIOHVBW-QBNMFFNISA-N
SMILES: COC1=CC=C2C(C(O[C@@]23CC[C@@H](C(N(CCN4CCCCC4)C)=O)CC3)=O)=C1
Biological Activity: H3R antagonist 5 (Compound 1b) is a selective histamine H3 receptor inverse agonist with a IC50 of 0.54 nM and the ability to cross the blood-brain barrier. H3R antagonist 5 can be used in central nervous system-related research[1].
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H3R antagonist 5 | H3R antagonist 5 (Compound 1b) is a selective histamine H3 receptor inverse agonist with a IC50 of 0.54 nM and the ability to cross the blood-brain barrier. H3R antagonist 5 can be used in central nervous system-related research. | |||||||||||||||||||||
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References
Keywords
