Picenadol
Picenadol (LY-150720) is an opioid mixed agonist-antagonist analgesic. Picenadol is an external racemic mixture, where its d-isomer (LY136596) is a potent μ-opioid receptor agonist, and the l-isomer (LY136595) is a weak μ-receptor competitive antagonist, which can inhibit the agonist effect and reduce the risk of dependence. Picenadol has anticholinergic activity.
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- CAS. Nr.: 79201-85-7
- Formel: C16H25NO
- Molecular Weight:247.38
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Biologische Aktivität
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μ Opioid Receptor/MOR |
Chemical Information
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CAS. Nr. 79201-85-7
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Molecular Weight 247.38
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Formel C16H25NO
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SMILES
CCC[C@]1([C@@H](C)CN(CC1)C)C2=CC(O)=CC=C2
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Synonyms
LY-150720
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
[1]. Carter RB, et al. Effects of LY150720 (picenadol), a novel mixed-action opioid, on schedule-controlled responding in the squirrel monkey. Pharmacol Biochem Behav. 1984 Nov;21(5):779-86. [Content Brief]
[2]. Zimmerman DM, et al. Picenadol. Drug Alcohol Depend. 1985 Feb;14(3-4):381-401. [Content Brief]
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Picenadol Related Classifications
HY-106601 Related Classifications
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