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Cat. No.: HY-16729

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Relenopride

(Synonyms: YKP10811)

Relenopride is a agonist of novel potent 5-HT₄ receptor partial with weak binding to 5-HT 2B receptors (K_i = 31 nM).

For research use only. We do not sell to patients.

CAS No.: 1221416-43-8
Formula: C₂₄H₃₀ClFN₄O₄
Molecular Weight:492.97

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (265 KB)

Relenopride Chemical Structure

CAS No.: 1221416-43-8

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Quantity

Sample (0.1mg)

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(In Japan)

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Bioz

Biological Activity

Description

Relenopride is a agonist of novel potent 5-HT₄ receptor partial with weak binding to 5-HT 2B receptors (K_i = 31 nM)^[1].

IC₅₀ & Target

5-HT_2B Receptor

All 5-HT Receptor Isoforms :

Chemical Information

CAS No. 1221416-43-8
Molecular Weight 492.97
Formula C₂₄H₃₀ClFN₄O₄
SMILES

NC(O[C@H](C1=CC=C(C=C1)F)CCN(CC2)CCC2CNC(C3=C(C=C(C(Cl)=C3)N)OC)=O)=O
Synonyms

YKP10811
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (265 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Anna Zielińska, et al. Chronic abdominal pain in irritable bowel syndrome - current and future therapies. Expert Rev Clin Pharmacol. 2018 Jul;11(7):729-739. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Dilution Calculator

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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