LBG20304
LBG20304 (compound 2s) is a ligand for the homologous GluK5 receptor (IC50: 432 nM), more than 40-fold selective over the homologous GluK1-3 isoforms. Low doses of LBG20304 (<10 μM) have no agonist or antagonist functional response at heterologous GluK2/5 receptors, and at high doses (>10 μM), it exhibits low agonist activity in neuronal slices (rat).
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C19H18N4O5
- Peso molecular:382.37
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Descripciòn
IC50 & Target
IC50: 432 nM (GluK5)[1]
Chemical Information
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Peso molecular 382.37
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Fòrmula C19H18N4O5
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SMILES
O=C([C@H]1NC[C@H](N2N=NC=C2C3=CC=C4C=C(O)C=CC4=C3)[C@@H]1CC(O)=O)O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LBG20304 Related Classifications
HY-159584 Related Classifications
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