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Referencia número: HY-10051

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GR203040

Name: GR203040
Brand: MedChemExpress
SKU: HY-10051
Price: 370.00 USD
Availability: InStock
Rating: 5 (1 reviews)

GR203040 is an orally active NK₁ receptor antagonist with a pK_i of 10.3. GR203040 shows potent antiemetic activity.

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No. CAS: 168398-02-5
Fòrmula: C₂₀H₂₆Cl₂N₆O
Peso molecular:437.37

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

GR203040 Chemical Structure

No. CAS: 168398-02-5

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Descripciòn

GR203040 is an orally active NK₁ receptor antagonist with a pK_i of 10.3. GR203040 shows potent antiemetic activity^[1].

IC₅₀ & Target

pKi: 10.3 (NK₁ receptor)^[1]

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Chemical Information

No. CAS 168398-02-5
Peso molecular 437.37
Fòrmula C₂₀H₂₆Cl₂N₆O
SMILES

COC1=CC=C(N2N=NN=C2)C=C1CN[C@@H]3[C@H](C4=CC=CC=C4)NCCC3.[H]Cl.[H]Cl
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Ward P, et al. Discovery of an orally bioavailable NK1 receptor antagonist, (2S,3S)-(2-methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with potent antiemetic activity. J Med Chem. 1995 Dec 22;38(26):4985-92. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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GR203040

Ver todos los productos específicos de isoformas Neurokinin Receptor

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