4 Results for "

208169

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "208169" in MCE Product Catalog:

14
14 Publications Verification
Cat. No.: HY-15455
CAS No.: 162401-32-3
Purity:  99.98%
Synonyms: APTA-2217; BYK 20869; B9302-107
Research Areas:  

Inflammation/Immunology

Roflumilast (APTA-2217) is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDE4A4, PDE4B1, and PDE4B2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
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1
1 Cited Publications
Cat. No.: HY-15455S
CAS No.: 1398065-69-4
Synonyms: APTA-2217-d4; BYK 20869-d4; B9302-107-d4
Roflumilast-d4 is the deuterium labeled Roflumilast. Roflumilast is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDEA4, PDEB1, and PDEB2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells .
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Cat. No.: HY-15455R
CAS No.: 162401-32-3
Synonyms: APTA-2217 (Standard); BYK 20869 (Standard); B9302-107 (Standard)
Roflumilast (Standard) is the analytical standard of Roflumilast. This product is intended for research and analytical applications. Roflumilast (APTA-2217) is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDEA4, PDEB1, and PDEB2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
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Cat. No.: HY-15455S2
CAS No.: 1189992-00-4
Synonyms: APTA-2217-d3; BYK 20869-d3; B9302-107-d3
Roflumilast-d3 is deuterium labeled Roflumilast. Roflumilast is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDEA4, PDEB1, and PDEB2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
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