GIPR antagonist 1
GIPR antagonist 1 is a GIPR antagonist with an IC50 of 4.8 nM. GIPR antagonist 1 inhibits glucose-dependent insulinotropic polypeptide receptor signaling. GIPR antagonist 1 can be used for the research of type 2 diabetes and obesity.
For research use only. We do not sell to patients.
- CAS No.: 3059497-30-9
- Formula: C28H29FN4O4
- Molecular Weight:504.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
GIPR antagonist 1 (Compound 27) (10-100 nM, 6 h) antagonizes human GIPR and inhibits downstream cAMP production in a concentration‑dependent manner in CHO‑K1 cells stably expressing human GIPR[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3059497-30-9
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Molecular Weight 504.55
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Formula C28H29FN4O4
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SMILES
FC(C=C1NC(N2[C@H](CCC2)C(NC3=CC=C(C4=C(N=C(C=C4)C(O)=O)C)C=C3)=O)=O)=C(C=C1)C(C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GIPR antagonist 1 Related Classifications
HY-179332 Related Classifications
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