GLP-1R/GIPR agonist-2
GLP-1R/GIPR agonist-2 is a GIPR agonist. GLP-1R/GIPR agonist-2 potentiates GIP(1-42)-induced intracellular cAMP production in cells expressing human GIPR. GLP-1R/GIPR agonist-2 can be used for the research of type II diabetes mellitus.
For research use only. We do not sell to patients.
- CAS No.: 2766799-78-2
- Formula: C32H43Cl2FN2O2
- Molecular Weight:577.60
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
GLP-1R/GIPR agonist-2 (Example 1) (30 min) acts as a positive allosteric modulator of the human GIPR in HEK293 cells, with an EC50 of 11.9 nM and maximal potentiation equivalent to 101% of the positive control response[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2766799-78-2
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Molecular Weight 577.60
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Formula C32H43Cl2FN2O2
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SMILES
COC1=CC=C([C@H](N(CC2)C(C3=CC=C(C=C3)C(C)C)C)C)C2=C1C4=CC(NCC(C)C)=C(C(F)=C4)O.Cl.Cl
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GLP-1R/GIPR agonist-2 Related Classifications
HY-171302 Related Classifications
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