GPR120 Agonist 4
GPR120 Agonist 4 (example 1) is a GPR120 agonist，with the EC50 values of 1 μM and 0.35 μM for β-arrestin A and Calcium A. GPR120 Agonist 4 can be used for the research of type II diabetes mellitus.
For research use only. We do not sell to patients.
- CAS No.: 1628641-89-3
- Formula: C21H15ClF5NO3
- Molecular Weight:459.79
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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GPR120 1 μM (EC50) |
GPR120 Agonist 4 (example 1) (0.012-25 μM, 90 min) can activate GPR120 through recruitment of β-Arrestin in CHO-K1 GPR120 β-Arrestin cells[1].
GPR120 Agonist 4 (0.012-25 μM, 90 min) promotes the release of Ca2+ in HEK293 with human GPR120 clone, which verifies the activation effect of GPR120 Agonist 4 on GPR120[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
GPR120 Agonist 4 (1/3/10 mg/kg, i.p., 15/30/45/60/90 min) inhibits the glucose level of starvation mouse model in a dose-dependent manner[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1628641-89-3
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Molecular Weight 459.79
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Formula C21H15ClF5NO3
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SMILES
O=C(CCC1=CC(F)=C(C(F)=C1)OCC2=C(C(F)(F)F)C=CN2C3=CC=C(C=C3)Cl)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GPR120 Agonist 4 Related Classifications
HY-160628 Related Classifications
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