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Heterobivalent ligand-1

Heterobivalent ligand-1 (compound 26) is a heterobivalent ligand for the Adenosine A 2A-dopamine D 2 receptor heteromer (K_DB1 A_2AR=2.1 nM, K_DB1 D₂R= 0.13 nM).

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CAS No.: 2888568-58-7
Formula: C₈₇H₁₁₇FN₁₆O₂₁
Molecular Weight:1741.95

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

Heterobivalent ligand-1 Chemical Structure

CAS No.: 2888568-58-7

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Biological Activity

Description

Heterobivalent ligand-1 (compound 26) is a heterobivalent ligand for the Adenosine A 2A-dopamine D 2 receptor heteromer (K_DB1 A_2AR=2.1 nM, K_DB1 D₂R= 0.13 nM)^[1].

All Adenosine Receptor Isoforms :

All Dopamine Receptor Isoforms :

Chemical Information

CAS No. 2888568-58-7
Molecular Weight 1741.95
Formula C₈₇H₁₁₇FN₁₆O₂₁
SMILES

O=C(CN(CC(OC)=O)CC(NCCOCCOCCOCCOCCOCCNC(COC1=CC=C(CCCN2N=CC3=C2N=C(N)N4C3=NC(C5=CC=CO5)=N4)C=C1)=O)=O)NCCOCCOCCOCCOCCOCCNC(CCC(NC6=CC=C(CCN7CN(C8=CC=CC=C8)C9(CCN(CCCC(C%10=CC=C(F)C=C%10)=O)CC9)C7=O)C=C6)=O)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Pulido D, et al. Heterobivalent Ligand for the Adenosine A2A-Dopamine D2 Receptor Heteromer. J Med Chem. 2022;65(1):616-632. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
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Chemical Information
Purity & Documentation
References

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Heterobivalent ligand-1

All Adenosine Receptor Isoforms

All Dopamine Receptor Isoforms