Human enteropeptidase-IN-2
Human enteropeptidase-IN-2 (compound 1c) is a highly potent enteropeptidase inhibitor. Human enteropeptidase-IN-2 can be used for anti-obesity research.
For research use only. We do not sell to patients.
- CAS No.: 3031537-31-9
- Formula: C20H19F3N4O7
- Molecular Weight:484.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
IC50(initial): 540 nM (enteropeptidase)[1]
IC50(app): 30 nM (enteropeptidase)[1]
Human enteropeptidase-IN-2 (compound 1c) has inhibitory activity against enteropeptidase with IC50(initial)* of 540 nM and IC50(app)** of 30 nM[1].
(*IC50(initial) refers to the inhibitory activity of human enteropeptidase after 6 min of incubation with the enzyme, substrate, and compound.
**IC50(app) refers to the apparent IC50 value after 120 min of incubation with the enzyme, substrate, and compound.)
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3031537-31-9
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Molecular Weight 484.38
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Formula C20H19F3N4O7
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SMILES
NC(NC1=CC=C(C=C1)C(OC2=CC=C(CC(NCC(O)=O)=O)C=C2)=O)=N.OC(C(F)(F)F)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Human enteropeptidase-IN-2 Related Classifications
HY-147931 Related Classifications
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