Gidazepam
Based on 1 Customer Validation
Gidazepam is an agonist of GABA receptor channels (GABA RCs).
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度 : 98.05%
- CAS 番号: 129186-29-4
- 分子式: C17H15BrN4O2
- 分子量:387.23
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
IC50 & Target
GABA receptor[1]
体外実験
Gidazepam demonstrates considerably lower affinities to GABA RCs than phenazepam, 3-hydrozyphenazepam, and Br-nordiazepam. This is manifested in different values of the inhibition constant (Ki) of binding of a specific ligand of benzodiazepine receptors, diazepam. For Gidazepam, the Ki value is 2,200±50 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
体内実験
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 129186-29-4
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性状 Solid
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分子量 387.23
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分子式 C17H15BrN4O2
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Color White to off-white
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SMILES
O=C(NN)CN1C(CN=C(C2=CC=CC=C2)C3=CC(Br)=CC=C31)=O
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別名
Gidasepam; Hidazepam; Hydazepam
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
体外:
DMSO : 250 mg/mL (645.61 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (280 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.5824 mL | 12.9122 mL | 25.8244 mL | 64.5611 mL |
| 5 mM | 0.5165 mL | 2.5824 mL | 5.1649 mL | 12.9122 mL | |
| 10 mM | 0.2582 mL | 1.2912 mL | 2.5824 mL | 6.4561 mL | |
| 15 mM | 0.1722 mL | 0.8608 mL | 1.7216 mL | 4.3041 mL | |
| 20 mM | 0.1291 mL | 0.6456 mL | 1.2912 mL | 3.2281 mL | |
| 25 mM | 0.1033 mL | 0.5165 mL | 1.0330 mL | 2.5824 mL | |
| 30 mM | 0.0861 mL | 0.4304 mL | 0.8608 mL | 2.1520 mL | |
| 40 mM | 0.0646 mL | 0.3228 mL | 0.6456 mL | 1.6140 mL | |
| 50 mM | 0.0516 mL | 0.2582 mL | 0.5165 mL | 1.2912 mL | |
| 60 mM | 0.0430 mL | 0.2152 mL | 0.4304 mL | 1.0760 mL | |
| 80 mM | 0.0323 mL | 0.1614 mL | 0.3228 mL | 0.8070 mL | |
| 100 mM | 0.0258 mL | 0.1291 mL | 0.2582 mL | 0.6456 mL |
Gidazepam 関連分類
HY-U00315 関連分類
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