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Cat. No.: HY-19733S1

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Lumateperone-d₄ tosylate

(Synonyms: ITI-007-d₄)

Lumateperone-d₄ tosylate (ITI-007-d₄ tosylate) is the deuterium labeled Lumateperone tosylate (HY-19733). Lumateperone (ITI-007) tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia.

For research use only. We do not sell to patients.

Formula: C₃₈H₄₀D₄FN₃O₇S₂
Molecular Weight:741.92

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Lumateperone-d₄ tosylate Chemical Structure

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vitro
- Application
Chemical Information
Purity & Documentation
Calculators
Help & FAQs
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Bioz

Biological Activity

Description

All 5-HT Receptor Isoforms :

All Dopamine Receptor Isoforms :

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

Unlabeled Cas 1187020-80-9
Molecular Weight 741.92
Formula C₃₈H₄₀D₄FN₃O₇S₂
SMILES

O=S(O)(C1=CC=C(C=C1)C)=O.CN2C3=C4C([C@@]5([H])[C@@](CCN(C5)CCCC(C6=C([2H])C([2H])=C(C([2H])=C6[2H])F)=O)([H])N4CC2)=CC=C3.O=S(O)(C7=CC=C(C=C7)C)=O
Synonyms

ITI-007-d₄
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.