1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. GABA Receptor
  3. mGAT3/4-IN-2

mGAT3/4-IN-2 

Cat. No.: HY-146281
Handling Instructions

mGAT3/4-IN-2 (compound 27b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.44 and 5.25, respectively.

For research use only. We do not sell to patients.

mGAT3/4-IN-2 Chemical Structure

mGAT3/4-IN-2 Chemical Structure

CAS No. : 2556833-68-0

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Description

mGAT3/4-IN-2 (compound 27b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.44 and 5.25, respectively[1].

IC50 & Target

pIC50: 5.12 ± 0.08 (mGAT1), 5.14 ± 0.07 (mGAT2), 5.44 ± 0.08 (mGAT3), 5.25 ± 0.04 (mGAT4)[1]

Molecular Weight

502.13

Formula

C26H32ClN3OS2

CAS No.
SMILES

CC1=C(SC=C1)/C(C2=C(C=CS2)C)=C\CCN(C(C(NCC3=C(C=CC=C3)Cl)=O)CCN)C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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mGAT3/4-IN-2
Cat. No.:
HY-146281
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