Synthesis of diprotected monosubstituted hydrazine derivatives from tert-butyl carbazates and boronic acids

  • Org Lett. 2003 Oct 30;5(22):4129-31. doi: 10.1021/ol035544v.
George W Kabalka  1 Sankar K Guchhait
Affiliations
  • 1. Departments of Chemistry and Radiology, The University of Tennessee, Knoxville, Tennessee 37996, USA. [email protected]
Abstract

[reaction: see text]. Diprotected monosubstituted hydrazine derivatives have been prepared via the reaction of tert-butyl carbazates with boronic acids catalyzed by cuprous chloride at room temperature.

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