S(-)-Cyanopindolol hemifumarate
S(−)-Cyanopindolol hemifumarate is an isomer of Cyanopindolol (HY-W795507). S(-)-Cyanopindolol hemifumarate is a 5-HT1A/1B serotonin receptor antagonist and a β3-adrenoceptor antagonist.
For research use only. We do not sell to patients.
- CAS No.: 874882-72-1
- Formula: C16H21N3O2·1/2C4H4O4
- Molecular Weight:345.20
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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β3 adrenoceptor |
5-HT1A Receptor |
5-HT1B Receptor |
Chemical Information
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CAS No. 874882-72-1
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Molecular Weight 345.20
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Formula C16H21N3O2·1/2C4H4O4
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SMILES
OC(/C=C/C(O)=O)=O.CC(C)(C)NC[C@H](O)COC1=C2C(NC(C#N)=C2)=CC=C1.[1/2]
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Giles H, et al. Characterization of a 5-HT1B receptor on CHO cells: functional responses in the absence of radioligand binding. Br J Pharmacol. 1996 Mar;117(6):1119-26. [Content Brief]
[2]. Hoey AJ, et al. Characteristics of cyanopindolol analogues active at the beta 3-adrenoceptor in rat ileum. Br J Pharmacol. 1996 Oct;119(3):564-8. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)