Sakamototide substrate peptide TFA

Name: Sakamototide substrate peptide TFA
Brand: MedChemExpress
SKU: HY-P1797A
Rating: 4.5 (1 reviews)

Cat. No.: HY-P1797A Purity: 98.79%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Sakamototide substrate peptide TFA is a peptide substrate for members of the AMPK family of kinases, used in kinase activity assays.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

Sakamototide substrate peptide TFA Chemical Structure

Size	Price	Stock	Quantity
Solid + Solvent
10 mM * 1 mL in Water ready for reconstitution	USD 714	In-stock	Estimated Time of Arrival: December 31
Solution
10 mM * 1 mL in Water	USD 714	In-stock	Estimated Time of Arrival: December 31
Solid
5 mg	USD 220	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 350	In-stock	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

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This product is a controlled substance and not for sale in your territory.

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Based on 1 publication(s) in Google Scholar

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Biological Activity
Purity & Documentation
References
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Description

Sakamototide substrate peptide TFA is a peptide substrate for members of the AMPK family of kinases, used in kinase activity assays^[1]^[2].

Molecular Weight

1853.92

Formula

C₇₁H₁₂₃F₃N₃₀O₂₅

Appearance

Solid

Color

White to off-white

Sequence

Ala-Leu-Asn-Arg-Thr-Ser-Ser-Asp-Ser-Ala-Leu-His-Arg-Arg-Arg

Sequence Shortening

ALNRTSSDSALHRRR

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Sealed storage, away from moisture

Powder	-80°C	2 years
	-20°C	1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

H₂O : 100 mg/mL (53.94 mM; Need ultrasonic)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	0.5394 mL	2.6970 mL	5.3940 mL
5 mM	0.1079 mL	0.5394 mL	1.0788 mL
10 mM	0.0539 mL	0.2697 mL	0.5394 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

Molarity Calculator
Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

In Vivo:

For the following dissolution methods, please prepare the working solution directly. It is recommended to prepare fresh solutions and use them promptly within a short period of time.
The percentages shown for the solvents indicate their volumetric ratio in the final prepared solution. If precipitation or phase separation occurs during preparation, heat and/or sonication can be used to aid dissolution.

Protocol 1

Add each solvent one by one: PBS
Solubility: 50 mg/mL (26.97 mM); Clear solution; Need ultrasonic

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

This product has good water solubility, please refer to the measured solubility data in water/PBS/Saline for details.

The concentration of the stock solution you require exceeds the measured solubility. The following solution is for reference only.If necessary, please contact MedChemExpress (MCE).

Purity & Documentation

Purity: 98.79%

Select Batch:

Data Sheet (269 KB) SDS (252 KB)

COA (241 KB) RP-HPLC (237 KB) Elemental Analysis Report (101 KB)

Handling Instructions (2659 KB)

References

[1]. Banerjee S,et al. Characterization of WZ4003 and HTH-01-015 as selective inhibitors of the LKB1-tumour-suppressor-activated NUAK kinases. Biochem J. 2014 Jan 1;457(1):215-25. [Content Brief]

[2]. Banerjee S, et al. Interplay between Polo kinase, LKB1-activated NUAK1 kinase, PP1βMYPT1 phosphatasecomplex and the SCFβTrCP E3 ubiquitin ligase. Biochem J. 2014 Jul 15;461(2):233-45. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

H₂O	1 mM	0.5394 mL	2.6970 mL	5.3940 mL	13.4849 mL
	5 mM	0.1079 mL	0.5394 mL	1.0788 mL	2.6970 mL
	10 mM	0.0539 mL	0.2697 mL	0.5394 mL	1.3485 mL
	15 mM	0.0360 mL	0.1798 mL	0.3596 mL	0.8990 mL
	20 mM	0.0270 mL	0.1348 mL	0.2697 mL	0.6742 mL
	25 mM	0.0216 mL	0.1079 mL	0.2158 mL	0.5394 mL
	30 mM	0.0180 mL	0.0899 mL	0.1798 mL	0.4495 mL
	40 mM	0.0135 mL	0.0674 mL	0.1348 mL	0.3371 mL
	50 mM	0.0108 mL	0.0539 mL	0.1079 mL	0.2697 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Sakamototide substrate peptideOthersInhibitorinhibitorinhibit

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Sakamototide substrate peptide TFA

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