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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
5 Results for "
ATPA
" in MedChemExpress (MCE) Product Catalog:
Products (5)
5 Results for "ATPA" in MCE Product Catalog:
Target:
Research Areas:
ATPA is a selective glutamate receptor GluR5 activator with EC50s of 0.66, 9.5, 1.4, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S741M), GluR5(S721T), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V), respectively .
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1 Cited Publications
Cat. No.: HY-P86665
Synonyms: ATP1A1; alpha 1 Sodium Potassium ATPAse; A1A1; AT1A1; AT1A1_HUMAN; ATPA-1; ATPAse Na+/K+transporting alpha 1 polypeptide; ATPAse Na+/K+transporting subunit alpha 1; BC010319; EC 3.6.3.9; MGC3285; MGC38419; MGC51750; Na K ATPAse alpha A catalytic polypeptide; Na K ATPAse catalytic subunit alpha A protein; Na(+)/K(+) ATPAse 1; Na(+)/K(+) ATPAse alpha-1 subunit; Na+, K+ATPAse alpha subunit; Na+/K+ATPAse alpha 1 subunit; Na+/K+ATPAse 1; Na, K ATPAse alpha 1 subunit; Nkaa1b; Sodium potassium ATPAse alpha 1 polypeptide; Sodium pump 1; Sodium pump subunit alpha-1; sodium-potassium ATPAse catalytic subunit alpha-1; Sodium/potassium-transporting ATPAse subunit alpha-1.
Synonyms: ACET
Target:
Research Areas:
UBP316 (ACET) is a highly potent and selective kainate receptor GluK1 (GluR5) antagonist, with a Kb value of 1.4 nM. UBP316 is effective at blocking the depression of both field excitatory postsynaptic potentials (fEPSPs) and monosynaptically-evoked GABAergic transmission induced by ATPA, a GluK1 selective agonist .
Cat. No.: HY-CE01941
Synonyms: Thio-ATPA-coenzyme A
Target:
Research Areas:
Thio-ATPA-CoA (Thio-ATPA-coenzyme A) is a coenzyme A derivative .
Cat. No.: HY-107605
CAS No.: 745055-86-1
Target:
Research Areas:
UBP296 is a potent and selective antagonist of GLUK5-containing kainate receptor in the spinal cord. UBP296 reversibly blocks ATPA-induced depressions of synaptic transmission, and affects AMPA receptor-mediated synaptic transmission directly in rat hippocampal slices .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
