3 Results for "

CGP62221

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "CGP62221" in MCE Product Catalog:

Cat. No.: HY-129491
CAS No.: 740816-86-8
Purity:  97.08%
Synonyms: CGP62221; O-Desmethyl PKC412
Target:  

PKC

Research Areas:  

Cancer

O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism. O-Desmethyl Midostaurin can be used as an indicator for Midostaurin metabolism in vivo . Midostaurin is a multi-targeted protein kinase inhibitor with IC50 ranging from 22-500 nM.
loading...
    loading...
Cat. No.: HY-W751181
Synonyms: CGP62221-13C6; O-Desmethyl PKC412-13C6
O-Desmethyl midostaurin- 13C6 (CGP62221- 13C6; O-Desmethyl PKC412- 13C6) is the 13C-labeled O-Desmethyl Midostaurin (HY-129491). O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism. O-Desmethyl Midostaurin can be used as an indicator for Midostaurin metabolism in vivo . Midostaurin is a multi-targeted protein kinase inhibitor?with?IC50?ranging from 22-500 nM.
loading...
    loading...
Cat. No.: HY-129491S
CAS No.: 2699608-28-9
Synonyms: CGP62221-d5; O-Desmethyl PKC412-d5
O-Desmethyl Midostaurin-d5 is a deuterium labeled O-Desmethyl PKC412. O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism .
loading...
    loading...