2. Others Metabolic Enzyme/Protease
  3. Isotope-Labeled Compounds Drug Metabolite
  4. O-Desmethyl Midostaurin-d5

O-Desmethyl Midostaurin-d5  (Synonyms: CGP62221-d5; O-Desmethyl PKC412-d5)

Cat. No.: HY-129491S
Handling Instructions

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O-Desmethyl Midostaurin-d5 is a deuterium labeled O-Desmethyl PKC412. O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism[1].

For research use only. We do not sell to patients.

O-Desmethyl Midostaurin-d<sub>5</sub> Chemical Structure

O-Desmethyl Midostaurin-d5 Chemical Structure

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Other Forms of O-Desmethyl Midostaurin-d5:

O-Desmethyl Midostaurin-d5 Related Antibodies

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Description

O-Desmethyl Midostaurin-d5 is a deuterium labeled O-Desmethyl PKC412. O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism[1].

IC50 & Target

IC50: active metabolite of Midostaurin[1]
Molecular Weight

561.64

Formula

C34H23D5N4O4
SMILES

O=C1C2=C(C(C3=C4C=CC=C3)=C5N4[C@]6(O[C@@H](N7C5=C2C8=C7C=CC=C8)C[C@H]([C@H]6O)N(C(C(C([2H])=C9[2H])=C(C([2H])=C9[2H])[2H])=O)C)C)CN1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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O-Desmethyl Midostaurin-d5 Related Classifications

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  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

O-Desmethyl Midostaurin-d5CGP62221-d5O-Desmethyl PKC412-d5Isotope-Labeled CompoundsDrug MetaboliteMetaboliteMidostaurincytochrome P450deuterium labeledInhibitorinhibitorinhibit

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