5 Results for "

GHS1a

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "GHS1a" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-19884B
CAS No.: 2863659-22-5
Synonyms: RM-131 TFA; BIM-28131 TFA
Target:  

GHSR

Research Areas:  

Metabolic Disease

Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin TFA is centrally penetrant. Relamorelin TFA increases growth hormone levels and accelerates gastric emptying. Relamorelin TFA has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research [1] .
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Cat. No.: HY-113906A
CAS No.: 1092476-84-0
Purity:  99.40%
Target:  

GHSR

Research Areas:  

Metabolic Disease

(αR,8aS)-GSK1614343 is the isomer of GSK1614343 (HY-113906). GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors [1].
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Cat. No.: HY-19884
CAS No.: 661472-41-9
Synonyms: RM-131; BIM-28131
Target:  

GHSR

Research Areas:  

Metabolic Disease

Relamorelin (RM-131), a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin is centrally penetrant. Relamorelin increases growth hormone levels and accelerates gastric emptying. Relamorelin has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research [1] .
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Cat. No.: HY-113906
CAS No.: 1092076-04-4
Target:  

GHSR

Research Areas:  

Metabolic Disease

GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors. GSK1614343 inhibits the calcium response induced by ghrelin with a pIC50 value of 7.90. GSK1614343 represents a useful tool to investigate the physiological relevance of the ghrelin system in rat models [1].
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Cat. No.: HY-19884A
CAS No.: 1809080-14-5
Synonyms: RM-131 acetate; BIM-28131 acetate
Target:  

GHSR

Research Areas:  

Metabolic Disease

Relamorelin (RM-131) acetate, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin acetate is centrally penetrant. Relamorelin acetate increases growth hormone levels and accelerates gastric emptying. Relamorelin acetate has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research [1] .
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