2 Results for "

KRAS dimerization

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "KRAS dimerization" in MCE Product Catalog:

Cat. No.: HY-139186
CAS No.: 2984236-79-3
Purity:  99.15%
Target:  

PROTACs Ras

Research Areas:  

Cancer

PROTAC KRAS G12C degrader-1 is a Cereblon-based KRAS G12C PROTAC degrader. PROTAC KRAS G12C degrader-1 induces CRBN/ KRAS G12C dimerization and degrades GFP- KRAS G12C in reporter cells .
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Cat. No.: HY-185217
CAS No.: 2429876-60-6
Target:  

Ras

Research Areas:  

Cancer

PPI stabilizer-1-1 (Compound 2) is a KRAS dimerizing agent. PPI stabilizer-1-1 dimerizes KRAS with a KD of 3.8 µM. PPI stabilizer-1-1 co-crystallizes with GCP-KRAS G12D. PPI stabilizer-1 can be used for the research of KRAS-driven cancers .
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