2 Results for "

Spiro-duocarmycin

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Spiro-duocarmycin" in MCE Product Catalog:

Cat. No.: HY-160969
CAS No.: 1642147-15-6
Research Areas:  

Cancer

Spiro-duocarmycin is a DNA minor groove N3-adenine alkylating agent. Spiro-duocarmycin exerts cytotoxic effects via DNA alkylation. Spiro-duocarmycin is the active spirocyclized form of seco-DUBA, which is incorporated as an inactive prodrug into the linker-drug construct of antibody-drug conjugates (ADCs). DUBA serves as an ADC payload that can be conjugated with monoclonal antibodies to synthesize antibody-drug conjugates (ADCs) .
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Cat. No.: HY-P1193
CAS No.: 129623-01-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

GR 82334 is a potent and specific reversible tachykinin NK1 receptor antagonist . GR 82334 inhibits substance P-induced sensitization by blocking SP NK1 receptors in naked mole-rats .
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