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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
8 Results for "
neurokinin 3 receptor
" in MedChemExpress (MCE) Product Catalog:
Products (8)
8 Results for "neurokinin 3 receptor" in MCE Product Catalog:
5
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Research Areas:
Fezolinetant is an antagonist of the neurokinin 3 receptor (NK3R), used for the treatment of menopausal hot flushes.
3
3 Cited Publications
Synonyms: MLE-4901; AZD2624; AZD4901
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Research Areas:
Pavinetant (MLE-4901) is a neurokinin-3 receptor (NK3R) antagonist.
Cat. No.: HY-117380
CAS No.: 224961-34-6
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SB 235375 is a potent and selective antagonist of the human neurokinin-3 (hNK-3) receptor designed by optimizing the structure of 2-phenyl-4-quinolinecarboxylic acid amide. SB 235375 displays high affinity for the hNK-3 receptor, with significantly higher binding affinities than hNK-2 and hNK-1 receptors. In vitro studies demonstrated its ability to block NK-3 receptor-mediated contraction and calcium mobilization, while in vivo, SB 223412 demonstrated oral and intravenous activity against NK-3 receptor-driven responses in animal models .
Cat. No.: HY-P3862
CAS No.: 110880-53-0
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Cat. No.: HY-P1588
CAS No.: 112748-19-3
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Cat. No.: HY-14432R
CAS No.: 941690-55-7
Synonyms: MLE-4901 (Standard); AZD2624 (Standard); AZD4901 (Standard)
Research Areas:
Pavinetant (Standard) is the analytical standard of Pavinetant. This product is intended for research and analytical applications. Pavinetant (MLE-4901) is a neurokinin-3 receptor (NK3R) antagonist.
Cat. No.: HY-181682
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Research Areas:
NK3R antagonist-1 is an orally active neurokinin-3 receptor (NK3R) antagonist with an IC50 of 53.61 nM. NK3R antagonist-1 reduces plasma luteinizing hormone (LH) levels in ovariectomized rat models. NK3R antagonist-1 is applicable to research related to menopausal hot flushes .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
