Talibegron hydrochloride
Based on 1 Customer Validation
Talibegron hydrochloride (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect.
For research use only. We do not sell to patients.
- Purity: 99.63%
- CAS No.: 178600-17-4
- Formula: C18H22ClNO4
- Molecular Weight:351.82
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Storage:
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
Talibegron hydrochloride (ZD2079 hydrochloride; 0.01-1000 μM) produces a concentration-dependent relaxation of phenylephrine-preconstricted isolated mesenteric arteries and causes full relaxation with 1 mM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 178600-17-4
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Appearance Solid
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Molecular Weight 351.82
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Formula C18H22ClNO4
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Color White to off-white
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SMILES
O=C(O)CC1=CC=C(OCCNC[C@H](O)C2=CC=CC=C2)C=C1.[H]Cl
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Synonyms
ZD2079 hydrochloride
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
-20°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvent & Solubility
DMSO : 125 mg/mL (355.30 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (268 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.8424 mL | 14.2118 mL | 28.4236 mL | 71.0591 mL |
| 5 mM | 0.5685 mL | 2.8424 mL | 5.6847 mL | 14.2118 mL | |
| 10 mM | 0.2842 mL | 1.4212 mL | 2.8424 mL | 7.1059 mL | |
| 15 mM | 0.1895 mL | 0.9475 mL | 1.8949 mL | 4.7373 mL | |
| 20 mM | 0.1421 mL | 0.7106 mL | 1.4212 mL | 3.5530 mL | |
| 25 mM | 0.1137 mL | 0.5685 mL | 1.1369 mL | 2.8424 mL | |
| 30 mM | 0.0947 mL | 0.4737 mL | 0.9475 mL | 2.3686 mL | |
| 40 mM | 0.0711 mL | 0.3553 mL | 0.7106 mL | 1.7765 mL | |
| 50 mM | 0.0568 mL | 0.2842 mL | 0.5685 mL | 1.4212 mL | |
| 60 mM | 0.0474 mL | 0.2369 mL | 0.4737 mL | 1.1843 mL | |
| 80 mM | 0.0355 mL | 0.1776 mL | 0.3553 mL | 0.8882 mL | |
| 100 mM | 0.0284 mL | 0.1421 mL | 0.2842 mL | 0.7106 mL |
Talibegron hydrochloride Related Classifications
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