Telotristat besilate
Telotristat besilate is a potent tryptophan hydroxylase inhibitor with an in vivo IC50 of 0.028 μM.
For research use only. We do not sell to patients.
- CAS No.: 1374745-52-4
- Formula: C31H28ClF3N6O6S
- Molecular Weight:705.10
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Protocols
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
Clinical Trial
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1374745-52-4
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Molecular Weight 705.10
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Formula C31H28ClF3N6O6S
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SMILES
N[C@H](C(O)=O)CC1=CC=C(C=C1)C2=NC(N)=NC(O[C@@H](C(F)(F)F)C3=CC=C(C=C3N4N=C(C=C4)C)Cl)=C2.O=S(C5=CC=CC=C5)(O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Telotristat besilate Related Classifications
HY-13055E Related Classifications
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